Cilostazol

Product Name: Cilostazol
Synonyms: 6-[4-(1-CYCLOHEXYL-1H-TETRAZOL-5-YL)BUTOXY]-3,4-DIHYDRO-2(1H)-QUINOLINONE;6-[4-(1-cyclohexyl-1h-tetrazol-5-yl)butoxy]-3,4-dihydro-2(1h)-quinolinone additional name: 6-[4-(1-cyclohexyl-5-tetrazolyl)butoxy]-1,2,3,4- tetrahydro-2-oxoquinolinone;CILASTAZOL;CILOSTAZOL;CILOSTAZOLE;RETAL;OPC 13013;OPC 21
CAS: 73963-72-1
MF: C20H27N5O2
MW: 369.46
Product Categories: Active Pharmaceutical Ingredients;Intermediates & Fine Chemicals;Pharmaceuticals;API’s;inhibitor;Cardiovascular APIs
mp 159-160°C
storage temp. Store at RT
solubility DMSO: 18 mg/mL, soluble
form solid
color off-white
Chemical Properties Colourless Needles
Usage A potent phosphodiesterase III A (PDE3A) inhibitor (IC50=0.2uM) and inhibitor of adenosine uptake. Has antimitogeni, antithrombotic, vasodilatory and cardiotonic properties in vivo. Also affects lipid levels in vivo
Usage antibacterial; LD50(iv) 280mg/kg(mouse).

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